Originally, Gestrinone was not exactly an anabolic androgenic steroid, or least it didn't start out that way.
Back in the 1970s, the drug was developed as an oral contraceptive!
However, it never made it past clinical trials and interest in it basically fizzled out.
In the 1980s it was determined that it had a number of androgenic properties, but it also came with estrogenic, progestational, and oddly enough, anti-estrogenic and anti-progestational capabilities.
At this point, Gestrinone was modified and synthesized into tetrahydrogestrinone, more commonly known today as THG.
THG is a designer steroid, and it is the more common term for formally known Gestrinone decades ago. Buy legal steroids online here.
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Even today, Gestrinone (also known as Nemestran, Dimetriose, Dimetrose, C21H24O2) is not particularly popular as an anabolic androgenic steroid.
Today, it might be used in the treatment of endometriosis. onclick=”ga(‘send’, ‘event’, ‘contextual’, ‘internal’, ‘contextual’, 5);”>Danazol is another that might be used.
A derivative of norethisterone (17α -ethynyl- 19-nortestosterone), it’s an oral drug that, through its mechanism of action, can inhibit gonadotropins released by the pituitary gland.
What good is it to bodybuilders? In its basic form, not much at all.
It’s the THG structure that even brings this substance to the attention of a bodybuilder or athlete.
This is because THG is strongly related to not only Gestrinone, along with its potentials, but also Trenbolone, an anabolic androgenic steroid that has the reputation of being one of the most potent anabolic androgenic steroids used by bodybuilders today.
It doesn’t seem to matter to bodybuilders that Trenbolone is an animal or veterinary grade steroid that is not intended for human use.
Nevertheless, the dangers of designer steroids are obvious to most experienced bodybuilders: unknown ingredients, untested results, unexpected side effects, and so forth.
A number of bodybuilders and athletes believe that THG is available over the counter, but it is not.
THG, as mentioned, is most commonly linked to Trenbolone and Gestrinone as so comparisons are often made between the two.
Before even considering usage, be aware that THG has not undergone many studies in regard to benefits or potentially dangerous side effects or adverse reactions in humans.
Bodybuilders do look for steroids that promote anabolic potential, but with reduced androgenic properties.
Androgens are responsible for the development of secondary sex male characteristics, but they do convert from testosterone into estrogen, in a process known as aromatization.
For men, this can mean:
For women, it can mean virilism.
Before taking any type of anabolic androgenic steroid, it’s important to anticipate side effects or unexpected adverse reactions.
Don’t just consider the benefits.
The same applies to Gestrinone implants, pills, or injections.
As well as to any drug or substance that is designed to mimic the effects of an anabolic androgenic steroid,
Risks increase when bodybuilders combine components like THG with other compounds like human growth hormone or some types of testosterone (at high doses).
While this may improve size as well as strength gains, it can also increase side effects.
Because THG is similar in nature to Trenbolone, it stands to reason that some of its side effects may be similar. However, Trenbolone and Gestrinone affect the body differently – as well as genders.
As mentioned, Gestrinone is basically an anti-progestin and anti-estrogenic steroid that is used to treat “female problems” such as endometriosis. It is also known to increase the potential for weight gain.
Some women experience virilism or male-type side effects with its use, which can include but are not limited to:
This is just the beginning. For men, one of the most common side effects of most anabolic androgenic steroids including this one is the suppression of endogenous or body-produced testosterone.
Because it’s an oral drug, the potential for liver toxicity is also strong.
As far as many bodybuilders are concerned, the benefits of using THG are not due to its anabolic or androgenic potential.
It does have the potential to improve performance, as well as the belief that it can be difficult to detect.
However, testing methods have advanced to incredible degrees today, and many anti-drug and doping tests are becoming more adept at identifying designer steroids such as THG.
Gestrinone dosage will depend on what you’re using it for, but start at around 2.5mg twice weekly for Endometriosis, to 5-10mg per day for bodybuilding.
Athletes in the past few decades have succumbed to not only loss of medals, but their reputation, their careers, and their livelihoods because of use of banned substances.
Before even considering use of a product like Gestrinone or Trenbolone, or THG (the Clear), regardless of how it’s sold, be aware of the risk associated with its use.Tetrahydrogestrinone THG SteroidMethyltrienoloneMetribolone Methyl TrenBolasteroneAndrostenedioneGestrinoneHCG SteroidNorbolethoneDnp SteroidEsiclene FormeboloneDihydroboldenoneNorclostebol Acetate Anabol 4 19MiboleroneStenbolone AnatrofinCheque DropsDanazol SteroidFluoxymesterone