Testosterone injection shots are commonly prescribed to men diagnosed with low levels of testosterone.
It is not recommended for enhancing physical strength, muscle building, bodybuilding, performance, or enhancement.
But even though the medical community and lawmakers frown upon performance use of testosterone injections, physique builders make up a large segment of the consumer base.
Testosterone is perhaps the most frequently used steroid in the weight training underground.
The allure of powerful gains in muscle mass and strength continue to lead many to use this “gateway steroid.”
However, a growing number of bodybuilders, concerned about the risks and dangers of anabolic steroids, have opted to forgo testosterone injections in favour of safe and legal natural dietary supplements that seek to mimic the effects of the steroid.
Testo-Max promises moderate gains without the painful injection schedule of pinning testosterone. Buy Testo-Max online here.
Table of Contents
There is a wide variety of Testosterone injections available.
The main differentiating factor between different testosterone shots is the ester attached.
One testosterone injection is not significantly more powerful or less powerful than another. At their core, they are all just testosterone and will ultimately have the same effect on the body.
The ester attached does not influence the effects of the injection. It only serves to prolong the release window of the drug by extending the drug’s half-life.
The weight of the ester can affect the potency of the drug in the sense that there is less testosterone per ml of the injection as it accommodates the ester.
Testosterone suspension, which is not esterified, is held to be the most potent form of testosterone for this reason.
Still, the effects of testosterone suspension vs. testosterone propionate on the body are not different.
One simply has more milligrams of testosterone per ml of the injection than the other, and this can easily be solved by adjusting the dosage of the esterified drug.
Esters have considerable implications for how a bodybuilder will structure their cycle, as short-estered drugs require a higher frequency of shots to maintain optimal blood plasma levels of the steroid.
Two illustrate this point, we will provide an overview of the 3 most popular forms of injectable testosterone in the steroid market.
This is considered to be the most common, widely recognised and often used form of esterified testosterone because it has an extremely long half-life when compared to the other forms of Testosterone.
It also boasts of an extended period of release, thereby making it easier to use for injections for patient or performance-use when needed.
For instance, a comparison between Testosterone Enanthate and Testosterone Propionate reveals that the half-life of Testosterone Enanthate which is about 7 to 10 days, makes it a lot easier to be give to patients as injections twice a week.
Most bodybuilders say that Testosterone Propionate needs to be pinned every other day.
Because it allows for less regular injections, Testosterone Enanthate is believed to be a better option as performance enhancer for needle shy patients.
Although considered to be similar to Testosterone Enanthate, Testosterone Cypionate contains a different chemical composition.
It has a higher half-life compared to Enanthate of about 12 days.
Another significant different between Cypionate and Enanthate is in their origin, while Cypionate originated from America, Enanthate has its origin outside the shores of the United States.
They are equally common amongst steroid users, although it can be argued that Enanthate has a higher consumption rate than Cypionate.
The similarities between Enanthate and Cypionate are such that they could be used interchangeably.
The major advantage of Cypionate, like every other extended half-life esterified compound, is in its ease of usage.
Occupying the number three spot in terms of popularity is Testosterone Propionate.
It is the first form of testosterone to be developed.
Testosterone Propionate has an extended half-life of about 4 and half days in the body. This is significantly shorter than Enanthate and Cypionate.
Its shorter half-life day makes it suitable if a user wants to have more control over blood plasma levels of the drug. It is known to require an increase in the number of injections per week.
For athletes adverse to the pain and dangers of self-administering needles, this is not believed to be a good option.
It ranks behind Enanthate and Cypionate in terms of popularity largely owing to the number of injections required during a cycle.
Notwithstanding, Cypionate has its fans. It is just doesn’t rank as high as Cypionate and Enanthate.
Taking into consideration the various life spans of the different types of Testosterone esters, there are unofficial and anecdotal guidelines in bodybuilding circles for administrating so as to attain stable blood plasma levels in the body.
These are the common guidelines recommended by experienced PED users to individuals who want to pin testosterone for performance and physique enhancement.
Others intending to use them for TRT should follow the advise of their doctor who is responsible for overseeing their treatment.
In the case of using Testosterone for performance enhancement, the dosage and application is a lot different from TRT as it involves a frequent administration schedule.
Increase in size and strength are reliant on achieving steady, peak blood plasma levels. This is held to mitigate the occurrence of certain side effects.
Testosterone Enanthate and Cypionate have been established to have extended half-lives of between 10 to 12 days.
However, performance users take them once a week for performance enhancing purposes at minimum.
For optimal blood plasma levels, bodybuilders usually recommend the user split their total weekly dosage in half and administer it twice a week with equal distance between dosages.
Some are adverse to the pain and risks of injecting at this frequency. If this is the case, a user might inject a single dose a week.
Still, this is widely discouraged in bodybuilding communities as it can lead to unstable blood plasma levels which leads to a greater risk of certain side effects while undercutting enhanced performance results.
Blended forms of Testosterone like the Sustanon 250 make for an interesting point of reference.
They tend to be on the losing side when it comes to popularity among athletes and weight trainers.
Compared to the single esterified testosterones mentioned in this article, Sustanon is dominantly regarded to be a poor choice.
The major disadvantage is due to the lack of control over the release rate of the various testosterones in the blend.
The different esterified testosterones make scheduling the dosage of the drug quite complex and difficult to manage.
At any rate, the recommended level of Sustanon dosage among physique builders is at least once every 7 to 10 days. This is felt to be required to achieve peak performance. This is also in sharp contrast to recommendations of once every 3 weeks stipulated in medical guideline.
Others tend to favor dosing the Sustanon 250 blend once every 3 days. This is based on the short-esterified forms of Testosterone in the blend.
The frequency of dosage for any blended variant of Testosterone should be based on the ester that contains the highest amount when compared to other esters available in the blend.
If the ester with the highest concentration is a short-ester variant like Propionate, the dosage schedule can be planned in the same way that it would be planned when cycling the single Testosteron Propionate form.
To bodybuilders, grasping the concept of achieving stable blood plasma levels of performance hormones is a must to achieve maximum gains and minimal side effects.
A lot of injectable testosterone has undergone esterification, increasing the half-life and prolonging the release of the hormone.
But this doesn’t guarantee stable levels of the drug in the bloodstream.
Even long-estered testosterone shots (Decanoate, Enanthate, Cypionate) could lead to a sharp increase in blood plasma levels upon the removal of the esters.
To administer the proper dosage and maintain a stable blood plasma hormone level required for the testosterone to function optimally, bodybuilders have to consider a number of points.
First, it usually takes about 48 hours after administration for the blood level of any ester variant to peak in terms of blood levels.
This might be surprising as a lot of information on bodybuilder sites and forums, which state that long-estered Testosterone takes a longer amount of time to start working.
In fact, these esterified forms of Testosterone actually get to work soon after they are injected into the body.
The difference the ester makes is the extended length of time it takes to achieve a steady state of hormone blood plasma level.
Getting to this level takes a longer period of time to achieve with esters likes Cypionate and Enanthate.
We already know that the life of a Testosterone is increased as a result of esterification due to the amount of time that would be required for the hormones to be freed by the ester bound enzymes.
The level of solubility in fats that arise as a result of esterification also contributed to the release rate of the drug in a small way.
This is insignificant when compared to the resulting increase in life span that the process of breaking down enzymes in contained in the esters themselves causes.
Esters consist mainly of long-chain hydrocarbons. This leads to them being classified as fats which makes them lipophilic.
The implication of this is that whichever compound they undergo chemical bonding with also becomes lipophilic as well.
Injectable Testosterone is therefore lipophilic.
When you consider the fact that Testosterone and other steroids are essentially lipids themselves, esterification increases the hormone’s fat-solubility.
What happens after an injection is that the oil in which the hormone can be found forms a deposit inside the muscle tissue thereby causing the hormone to separate from the oil and enter the bloodstream.
Esters containing a long hydrocarbon chain would make the hormones more fat-soluble, and this would in turn lead to a prolonged period before the hormone is released into the body.
This can extend the half-life of steroids containing esters with long hydrocarbon chains like Deca-Durabolin. Sometimes traces can be found in fatty tissues in the body for months after it has been injected into the body.
When the hormone injected into the body has been released for circulation into the bloodstream, the enzymes get to work on breaking the esters from the hormones.
At this point the steroid hormones are still inactive and cannot carry out any function unless the ester has totally been removed from the hormone.
The difference in price between pharmaceutical and underground Testosterone could be significant.
However, many performance users report that this isn’t the case.
It should be noted that when compared to other high end anabolic steroids like Anavar and Primobolan, Testosterone is a lot cheaper to produce and distribute.
This means the price difference between the pharmaceutical grade steroids and the underground testosterone wouldn’t be as high as the others.
For example, the Pharmaceutical grade of Testosterone Enanthate goes for about $13 to $15 for 1ml vial which contains about 250mg per ml.
The underground grade price for the same product would be about $60 to $90 for a single ml vial which contains about 250mg/ml.
Assuming we were to carry out a comparative cost analysis we would find out that the pharmaceutical grade testosterone goes for about $0.052 to $0.06 per mg while the underground grade of Testosterone Enanthate goes for about $0.024 to $0.036 per mg.
For Testosterone Cypionate, the pharmaceutical grade goes for about $15 to $18 for 1ml vial which contains 250mg/ml while the underground lab grade goes for $60 to $90 which is the cost of a 10ml vial at 250mg/ml.
A comparative cost analysis reveals that the pharmaceutical grade testosterone goes for about $0.06 to $0.072 per mg while the underground grade of Testosterone Enanthate goes for about $0.024 to $0.036 per mg (which is the same amount as Testosterone Cypionate this is due to the similarity in the composition of both compounds).
In the case of Testosterone Propionate, the pharmaceutical grade goes for about $4 to $6 for 1ml vial which contains 50mg/ml while the underground lab grade goes for $45 to $65 which is the cost of a 10ml vial at 250mg/ml.
A comparative cost analysis reveals that the pharmaceutical grade testosterone goes for about $0.08 to $0.12 per mg while the underground grade of Testosterone Propionate goes for about $0.045 to $0.065 per mg.
For the Sustanon 250 blend, the pharmaceutical grade goes for about $6 – $15 for 1ml vial which contains 250mg/ml while the underground lab grade goes for $50 – $100 for a 10ml vial at 250mg/ml.
A comparative cost analysis reveals that the pharmaceutical grade testosterone goes for about $0.024 – $0.06 per mg while the underground grade of Sustanon 250 goes for about $0.02 – $0.04 per mg.
It is important to note that the price of the underground grade products could differ significantly due to the nature of the manufacturing process and a lack of regulation in place to monitor the production and distribution process.
Normal (average) testosterone levels in men range 270 or 300 to 1070 ng (nanograms) per deciliter.
Test can be bound to proteins known as sex hormone binding globulin or SHBG.
Free levels that are not bound to protein can measure anywhere from 50 to 210 pg/mL (picograms per milliliter).
Testosterone is a very powerful hormone normally produced in adequate levels by the testicles (testes glands), following instructions to do so by the pituitary gland.
The pituitary gland is one of many that make up the endocrine system and is responsible for overseeing all glands’ functions, including secretions.
The pituitary gland receives a signal hormone from the hypothalamus gland (both located deep in the brain) to boost synthesis or production of testosterone in the testes.
This signal hormone is called luteinizing hormone or LH.
In some men, low levels can be caused by some type of dysfunction or malfunction of either the pituitary or the hypothalamus glands in the brain.
Other factors may contribute to the need for injections such as medical conditions like kidney disease.
At the other end of the spectrum, higher than normal levels of testosterone may be caused by conditions like testicular cancer or cancer of the adrenal glands.
Some genetic conditions can also cause low testosterone levels including Down’s syndrome and Klinefelter syndrome.
Cirrhosis of the liver, treatments for cancers in the body as well as alcoholism can contribute to low testosterone levels.
A deficiency of the luteinizing hormone-releasing hormone gonadotropin caused by an injury or tumors to the pituitary or hypothalamus glands are also potential circumstances that result in low testosterone levels for which therapy may be recommended.
Because low T levels can be caused by a myriad of conditions, talk to your doctor about the safety of taking shots.
Injectable testosterone may provide some benefits in testosterone replacement therapies, but they are not effective for everyone, or may be associated with increased risks that outweigh benefits.
This is especially true for seniors.
Injections are prescription only.
(Of course, while a number of non-prescribed injectable testosterone solutions are available through Internet or other resources, they are not recommended).
Injections like Testosterone Cypionate are generally prescribed for the treatment of congenital or acquired primary hypogonadism.
Talk to your doctor about the safety and efficacy of treatments as well as different types of injections.
A number of pills and topical ointments are also available, but your doctor will determine which form or method of application such as topical testosterone versus or injectable is most likely to provide you with the benefits you’re looking for.
Side effects associated with testosterone injections range from mild and transitory to severe and sometimes even life-threatening.
Discuss potential side effects with your doctor.
If you notice any changes in your physical or mental status, discuss with your doctor, as dosages may need to be adjusted.
Testosterone Cypionate injections are classified as Schedule III controlled substances.
Minor side effects range from irritation at the injection site, headache, and skin changes to more severe adverse reactions that can impact numerous body systems.
Moderate to severe side effects that affect the nervous system can include:
Gastrointestinal system side effects can include but are not limited to nausea (sometimes with vomiting), allergic reactions, or inflammation and pain at the injection site.
Such complaints are relatively common. Male pattern baldness, seborrhea, and acne have also been reported.
Severe adverse reactions may also affect the cardiovascular system and initiate myocardial infarction (heart attack), stroke, or disturbances in electrolyte and fluid levels in the body that can negatively impact organs and system functions.
Blood clots (venous thromboembolism) have also been noted as has reduced clotting capabilities in individuals already being treated with anticoagulant therapies and medications such as Warfarin.
Numerous types of injectable testosterone can provide benefits for many men, but they also come with side effects for many.
Talk to your doctor about the safety and benefits of testosterone shots, and carefully weigh them against potential risks.
There are other options such as changing your diet and foods you eat.Testopel Implants PelletsTestopel Reviews CostTestopel Side EffectsTestosterone ImplantsTestosterone PelletsTestosterone Pellets for WomenTestosterone PrescriptionTestosterone Replacement TherapyTestosterone Injections for SaleTestosterone Injections ShotsTestosterone Injections Side EffectsTestosterone MedicationTestosterone Patch